SCHEMBL14938841

SCHEMBL14938841

CCc1cccc(C2(N3CCN(Cc4cccs4)CC3)C(=O)c3ccccc3C2=O)n1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
HSD17B10 Q99714 1/20 0.42
DRD4 P21917 9/20 0.41
DRD3 P35462 6/20 0.41
DRD2 P14416 4/20 0.40
HTT P42858 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
DRD5 P21918 3/20 0.37
CHRM2 P08172 1/20 0.36
CHRM3 P20309 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
PARP1 P09874 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940461 0.84 NPSR1 (0.62) NPSR1SMN1; SMN2HSD17B10DRD2ALDH1A1
SCHEMBL14939130 0.84 NPSR1 (0.47) NPSR1DRD4DRD3DRD2MAPT
SCHEMBL14939113 0.83 NPSR1 (0.53) NPSR1KDM4EALDH1A1PARP1
SCHEMBL14939131 0.81 KMT2A (0.46) NPSR1HTTKDM4EALDH1A1MAPT
SCHEMBL14940522 0.81 NPSR1 (0.53) NPSR1SMN1; SMN2HSD17B10DRD2HTT
SCHEMBL14939607 0.81 NPSR1 (0.53) NPSR1DRD4DRD2HTTKDM4E
SCHEMBL14939717 0.80 NPSR1 (0.46) NPSR1SMN1; SMN2HSD17B10HTTKDM4E
SCHEMBL14939434 0.80 NPSR1 (0.51) NPSR1HTTKDM4EALDH1A1MAPT
SCHEMBL14939834 0.79 NPSR1 (0.53) NPSR1DRD4DRD3DRD2KDM4E
SCHEMBL14939051 0.79 NPSR1 (0.50) NPSR1DRD2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed