SCHEMBL14939113

SCHEMBL14939113

CCc1cccc(C2(N3CCN(Cc4ccncc4)CC3)C(=O)c3ccccc3C2=O)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.53
KDM4E B2RXH2 5/20 0.39
ALDH1A1 P00352 2/20 0.38
TSHR P16473 4/20 0.38
OPRL1 P41146 1/20 0.38
MEN1 O00255 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP3A4 P08684 3/20 0.37
CYP2D6 P10635 3/20 0.37
CYP2C9 P11712 2/20 0.37
USP2 O75604 1/20 0.36
TP53 P04637 1/20 0.36
LSS P48449 1/20 0.36
TNKS O95271 1/20 0.36
PARP1 P09874 1/20 0.36
PARP10 Q53GL7 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
PARP4 Q9UKK3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940461 0.92 NPSR1 (0.62) NPSR1ALDH1A1TSHRMEN1MAPK1
SCHEMBL14939607 0.89 NPSR1 (0.53) NPSR1KDM4EALDH1A1MEN1MAPK1
SCHEMBL14940522 0.89 NPSR1 (0.53) NPSR1KDM4EALDH1A1TSHRMEN1
SCHEMBL14939051 0.87 NPSR1 (0.50) NPSR1
SCHEMBL14939834 0.87 NPSR1 (0.53) NPSR1KDM4EALDH1A1TSHRTP53
SCHEMBL14939130 0.86 NPSR1 (0.47) NPSR1MEN1KMT2ACYP2D6
SCHEMBL14939434 0.85 NPSR1 (0.51) NPSR1KDM4EALDH1A1MEN1KMT2A
SCHEMBL14939717 0.84 NPSR1 (0.46) NPSR1KDM4EALDH1A1MEN1KMT2A
SCHEMBL14938841 0.83 NPSR1 (0.43) NPSR1KDM4EALDH1A1PARP1
SCHEMBL14939131 0.83 KMT2A (0.46) NPSR1KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed