SCHEMBL14939008

SCHEMBL14939008

Cc1cccc(C2Cc3c(F)cccc3C2=O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 6/20 0.52
ALOX15 P16050 1/20 0.47
ALOX12 P18054 1/20 0.47
PBRM1 Q86U86 1/20 0.42
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ACHE P22303 1/20 0.39
SIRT2 Q8IXJ6 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
MAPT P10636 2/20 0.37
TP53 P04637 1/20 0.37
THRB P10828 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HSD17B10 Q99714 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPK1 P28482 1/20 0.36
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940296 0.90 CYP19A1 (0.41) CYP19A1ALOX15ALOX12PBRM1ACHE
SCHEMBL14939087 0.86 CYP19A1 (0.43) CYP19A1ALOX15ALOX12PBRM1TDP1
SCHEMBL14939611 0.85 CYP19A1 (0.55) CYP19A1L3MBTL1SIRT2MEN1KMT2A
SCHEMBL14940317 0.83 CYP19A1 (0.57) CYP19A1ACHEKMT2AMAPTTP53
SCHEMBL14939220 0.78 CYP19A1 (0.59) CYP19A1ALOX15ALOX12TDP1L3MBTL1
SCHEMBL14939388 0.76 CYP19A1 (0.48) CYP19A1ALOX15ALOX12TDP1L3MBTL1
SCHEMBL6472550 0.72 ACHE (0.66) CYP19A1ACHEMAPK1HTR2CNOS3
SCHEMBL4742707 0.71 ACHE (0.60) CYP19A1ACHEKMT2AMAPTTP53
SCHEMBL14939619 0.70 SLC6A2 (0.52) CYP19A1ALOX15ALOX12L3MBTL1ACHE
SCHEMBL16556014 0.70 ACHE (0.41) CYP19A1ACHEMAPK1HTR2CNOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed