SCHEMBL14940317

SCHEMBL14940317

O=C1c2cccc(F)c2CC1c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 9/20 0.57
HTR2B P41595 2/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
NOS3 P29474 1/20 0.39
NOS2 P35228 1/20 0.39
DRD2 P14416 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
CFTR P13569 1/20 0.37
GOPC Q9HD26 1/20 0.37
ACHE P22303 1/20 0.37
TSHR P16473 1/20 0.37
KMT2A Q03164 1/20 0.37
KIF11 P52732 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939611 0.86 CYP19A1 (0.55) CYP19A1HTR2BMAPK1NOS3NOS2
SCHEMBL14939008 0.83 CYP19A1 (0.52) CYP19A1TP53CYP3A4MAPTMAPK1
SCHEMBL14940296 0.81 CYP19A1 (0.41) CYP19A1MAPK1NOS3NOS2ACHE
SCHEMBL14939420 0.80 CYP19A1 (0.45) CYP19A1HTR2BLMNATP53CYP1A2
SCHEMBL5951729 0.80 CYP19A1 (0.45) CYP19A1HTR2BLMNATP53CYP1A2
SCHEMBL4742707 0.80 ACHE (0.60) CYP19A1HTR2BLMNATP53CYP1A2
SCHEMBL14939087 0.78 CYP19A1 (0.43) CYP19A1TP53NOS3NOS2ACHE
SCHEMBL1582845 0.78 CYP19A1 (0.43) CYP19A1HTR2BLMNATP53CYP1A2
SCHEMBL14939214 0.78 ACHE (0.62) CYP19A1LMNAMAPTACHE
SCHEMBL16556014 0.75 ACHE (0.41) CYP19A1HTR2BMAPK1NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed