SCHEMBL14939276

SCHEMBL14939276

COc1ccc(F)cc1CN1CCN(C2(c3ccccc3)C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.59
MAPT P10636 4/20 0.51
KMT2A Q03164 3/20 0.48
TACR1 P25103 2/20 0.46
DRD2 P14416 1/20 0.46
DRD4 P21917 1/20 0.46
HRH2 P25021 1/20 0.46
HRH1 P35367 1/20 0.46
DRD3 P35462 1/20 0.46
KDM4E B2RXH2 3/20 0.44
MEN1 O00255 2/20 0.44
TSHR P16473 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TP53 P04637 1/20 0.43
LMNA P02545 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939877 0.91 NPSR1 (0.47) NPSR1MAPTKMT2ATACR1DRD2
SCHEMBL14939174 0.90 NPSR1 (0.65) NPSR1MAPTKMT2AKDM4EMEN1
SCHEMBL14939418 0.87 NPSR1 (0.61) NPSR1MAPTKMT2ADRD2DRD4
SCHEMBL14939270 0.87 NPSR1 (0.61) NPSR1MAPTKMT2ADRD2DRD4
SCHEMBL14939013 0.87 NPSR1 (0.64) NPSR1MAPTKMT2ADRD2KDM4E
SCHEMBL14938779 0.85 NPSR1 (0.65) NPSR1MAPTKMT2AKDM4EMEN1
SCHEMBL14940325 0.84 NPSR1 (0.64) NPSR1MAPTKMT2ADRD4KDM4E
SCHEMBL14939775 0.84 NPSR1 (0.52) NPSR1MAPTKMT2AKDM4EMEN1
SCHEMBL14940046 0.83 NPSR1 (0.54) NPSR1MAPTKMT2AKDM4EMEN1
SCHEMBL14938962 0.83 NPSR1 (0.54) NPSR1MAPTKMT2AKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed