SCHEMBL14939877

SCHEMBL14939877

COc1ccc(F)cc1CN1CCN(C2(c3cc(C)cc(C)c3)C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.47
KMT2A Q03164 2/20 0.46
TACR1 P25103 2/20 0.44
TP53 P04637 1/20 0.43
KDM4E B2RXH2 3/20 0.42
TSHR P16473 1/20 0.42
CYP2D6 P10635 1/20 0.41
MAPT P10636 3/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
HSD17B10 Q99714 1/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
HRH2 P25021 1/20 0.41
HRH1 P35367 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939276 0.91 NPSR1 (0.59) NPSR1KMT2ATACR1TP53KDM4E
SCHEMBL14938988 0.90 KDM4E (0.52) NPSR1KMT2ATP53KDM4ETSHR
SCHEMBL14939990 0.89 KDM4E (0.51) NPSR1KMT2ATACR1TP53KDM4E
SCHEMBL14939842 0.89 NPSR1 (0.50) NPSR1KMT2ATP53KDM4EMAPT
SCHEMBL14939401 0.89 NPSR1 (0.50) NPSR1KMT2ATP53KDM4EMAPT
SCHEMBL14939859 0.87 TP53 (0.49) NPSR1KMT2ATP53KDM4ETSHR
SCHEMBL14939141 0.86 HTR7 (0.44) NPSR1KMT2ATACR1TP53KDM4E
SCHEMBL14939948 0.85 NPSR1 (0.48) NPSR1KMT2ATP53KDM4EMAPT
SCHEMBL14939857 0.85 NPSR1 (0.48) NPSR1KMT2ATP53KDM4EMAPT
SCHEMBL14939609 0.84 NPSR1 (0.52) NPSR1KMT2ATP53TSHRCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed