SCHEMBL14939288

SCHEMBL14939288

CCc1cccc(C2(N3CCN(Cc4ccccc4C)CC3)Cc3cc(C)ccc3C2=O)c1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.40
ALDH1A1 P00352 5/20 0.37
MEN1 O00255 5/20 0.37
KDM4E B2RXH2 2/20 0.37
GAA P10253 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 2/20 0.35
CYP2A13 Q16696 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HTR6 P50406 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940164 0.93 KMT2A (0.43) KMT2AALDH1A1MEN1KDM4EGAA
SCHEMBL14939708 0.90 KMT2A (0.42) KMT2AALDH1A1MEN1KDM4EGAA
SCHEMBL14940207 0.88 ALDH1A1 (0.46) KMT2AALDH1A1KDM4EGAANPSR1
SCHEMBL14938926 0.86 NPSR1 (0.38) KMT2AALDH1A1MEN1GAANPSR1
SCHEMBL14939089 0.86 KMT2A (0.42) KMT2AALDH1A1MEN1KDM4EGAA
SCHEMBL14939091 0.86 KMT2A (0.42) KMT2AALDH1A1MEN1KDM4EGAA
SCHEMBL14939559 0.86 KMT2A (0.42) KMT2AALDH1A1MEN1KDM4EGAA
SCHEMBL14938855 0.85 ALDH1A1 (0.38) KMT2AALDH1A1MEN1KDM4EGAA
SCHEMBL14940190 0.85 ALDH1A1 (0.37) KMT2AALDH1A1MEN1KDM4EGAA
SCHEMBL14939099 0.83 KMT2A (0.43) KMT2AALDH1A1MEN1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed