SCHEMBL14939708

SCHEMBL14939708

Cc1ccc2c(c1)CC(c1ccccc1)(N1CCN(Cc3ccccc3C)CC1)C2=O

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
NPSR1 Q6W5P4 2/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
ATM Q13315 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CYP2A13 Q16696 1/20 0.39
GRIN2B Q13224 1/20 0.39
LMNA P02545 2/20 0.38
ACHE P22303 1/20 0.38
RAB9A P51151 1/20 0.38
HTR6 P50406 1/20 0.38
COMT P21964 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939099 0.93 KMT2A (0.43) KMT2AALDH1A1KDM4ENPSR1MEN1
SCHEMBL14940207 0.90 ALDH1A1 (0.46) KMT2AALDH1A1KDM4ENPSR1GAA
SCHEMBL14939941 0.90 KMT2A (0.47) KMT2AALDH1A1KDM4ENPSR1MEN1
SCHEMBL14940048 0.90 ALDH1A1 (0.44) KMT2AALDH1A1KDM4ENPSR1MEN1
SCHEMBL14939288 0.90 KMT2A (0.40) KMT2AALDH1A1KDM4ENPSR1MEN1
SCHEMBL14939629 0.88 KMT2A (0.45) KMT2AALDH1A1KDM4ENPSR1MEN1
SCHEMBL14939400 0.88 NPSR1 (0.52) KMT2AALDH1A1KDM4ENPSR1MEN1
SCHEMBL14939559 0.88 KMT2A (0.42) KMT2AALDH1A1KDM4ENPSR1MEN1
SCHEMBL14939091 0.88 KMT2A (0.42) KMT2AALDH1A1KDM4ENPSR1MEN1
SCHEMBL14939089 0.88 KMT2A (0.42) KMT2AALDH1A1KDM4ENPSR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed