SCHEMBL14939295

SCHEMBL14939295

Cc1cc(C)cc(C2(N3CCN(Cc4cc(F)ccc4C)CC3)C(=O)c3cccc(F)c3C2=O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.40
ALDH1A1 P00352 3/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 2/20 0.36
TP53 P04637 1/20 0.36
LMNA P02545 1/20 0.35
BCHE P06276 1/20 0.34
ACHE P22303 1/20 0.34
KDM4E B2RXH2 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
HTT P42858 1/20 0.33
P2RX7 Q99572 1/20 0.33
HTR7 P34969 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
MEN1 O00255 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
CA1 P00915 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940114 0.93 NPSR1 (0.41) NPSR1ALDH1A1GAAMAPTLMNA
SCHEMBL14939343 0.91 NPSR1 (0.51) NPSR1ALDH1A1GAAMAPTTP53
SCHEMBL14939945 0.90 NPSR1 (0.44) NPSR1ALDH1A1GAAMAPTTP53
SCHEMBL14939842 0.90 NPSR1 (0.50) NPSR1ALDH1A1GAAMAPTTP53
SCHEMBL14939943 0.88 NPSR1 (0.41) NPSR1ALDH1A1MAPTTP53LMNA
SCHEMBL14939141 0.87 HTR7 (0.44) NPSR1ALDH1A1MAPTTP53LMNA
SCHEMBL14938747 0.87 NPSR1 (0.44) NPSR1ALDH1A1GAAMAPTTP53
SCHEMBL14939857 0.86 NPSR1 (0.48) NPSR1ALDH1A1GAAMAPTTP53
SCHEMBL14939673 0.86 NPSR1 (0.51) NPSR1ALDH1A1MAPTTP53LMNA
SCHEMBL14939053 0.85 NPSR1 (0.45) NPSR1ALDH1A1GAAMAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed