SCHEMBL14939334

SCHEMBL14939334

Cc1cnccc1C1(Br)C(=O)c2ccccc2C1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.49
ALDH1A1 P00352 4/20 0.41
RECQL P46063 3/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
TSHR P16473 2/20 0.41
ALOX12 P18054 2/20 0.41
MAPK1 P28482 1/20 0.41
CASP1 P29466 1/20 0.41
BACE1 P56817 1/20 0.41
EHMT2 Q96KQ7 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
POLB P06746 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
S100A4 P26447 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940453 0.79 CYP2D6 (0.62) CYP2D6ALDH1A1RECQLL3MBTL1CA1
SCHEMBL14939588 0.72 ALDH1A1 (0.50) CYP2D6ALDH1A1RECQLL3MBTL1CA1
SCHEMBL14938951 0.71 ALDH1A1 (0.45) CYP2D6ALDH1A1RECQLL3MBTL1CA1
SCHEMBL14939487 0.71 ALDH1A1 (0.45) CYP2D6ALDH1A1RECQLL3MBTL1CA1
SCHEMBL14939984 0.71 CYP2D6 (0.45) CYP2D6ALDH1A1RECQLL3MBTL1CA1
SCHEMBL14939595 0.70 KMT2A (0.44) CYP2D6ALDH1A1RECQLL3MBTL1CA1
SCHEMBL9434988 0.69 CYP2D6 (0.48) CYP2D6ALDH1A1RECQLCA1CA2
SCHEMBL14939676 0.69 CYP2D6 (0.42) CYP2D6ALDH1A1RECQLL3MBTL1CA1
SCHEMBL14939387 0.68 ALDH1A1 (0.45) CYP2D6ALDH1A1RECQLL3MBTL1CA1
SCHEMBL14939316 0.68 NPC1 (0.46) CYP2D6ALDH1A1RECQLL3MBTL1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed