SCHEMBL14939588

SCHEMBL14939588

O=C1c2ccccc2C(=O)C1(Br)c1ccncc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
TSHR P16473 2/20 0.50
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
ALOX12 P18054 2/20 0.50
CA7 P43166 2/20 0.50
RECQL P46063 2/20 0.50
CA9 Q16790 2/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
BACE1 P56817 2/20 0.50
EHMT2 Q96KQ7 2/20 0.50
MAPK1 P28482 1/20 0.50
CASP1 P29466 1/20 0.50
CYP2D6 P10635 1/20 0.44
MAPT P10636 4/20 0.41
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
NPC1 O15118 2/20 0.41
TP53 P04637 2/20 0.41
MAPK10 P53779 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939057 0.83 ALDH1A1 (0.52) ALDH1A1TSHRCA1CA2ALOX12
SCHEMBL14938951 0.79 ALDH1A1 (0.45) ALDH1A1TSHRCA1CA2ALOX12
SCHEMBL14939461 0.78 CA1 (0.46) ALDH1A1TSHRCA1CA2ALOX12
SCHEMBL14939402 0.76 CYP2D6 (0.49) ALDH1A1TSHRCA1CA2ALOX12
SCHEMBL14940123 0.76 ALDH1A1 (0.47) ALDH1A1TSHRCA1CA2ALOX12
SCHEMBL14939387 0.76 ALDH1A1 (0.45) ALDH1A1TSHRCA1CA2ALOX12
SCHEMBL14939550 0.75 KCNQ2 (0.44) ALDH1A1TSHRCA1CA2ALOX12
SCHEMBL14940028 0.73 CA1 (0.42) ALDH1A1TSHRCA1CA2ALOX12
SCHEMBL14939206 0.72 ALDH1A1 (0.45) ALDH1A1TSHRCA1CA2ALOX12
SCHEMBL14939984 0.72 CYP2D6 (0.45) ALDH1A1TSHRCA1CA2ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed