SCHEMBL14939362

SCHEMBL14939362

CN(C)c1nccc(C2(Br)C(=O)c3ccccc3C2=O)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.41
DYRK1A Q13627 11/20 0.39
DYRK3 O43781 1/20 0.37
CLK1 P49759 1/20 0.37
CLK2 P49760 1/20 0.37
CLK3 P49761 1/20 0.37
JAK3 P52333 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
PNCK Q6P2M8 1/20 0.37
HASPIN Q8TF76 1/20 0.37
DYRK2 Q92630 1/20 0.37
HIPK2 Q9H2X6 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
DYRK4 Q9NR20 1/20 0.37
STK39 Q9UEW8 1/20 0.37
WNK2 Q9Y3S1 1/20 0.37
DYRK1B Q9Y463 1/20 0.37
ALDH1A1 P00352 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939567 0.76 CYP2D6 (0.41) CYP2D6DYRK1AALDH1A1TSHRMAPK1
SCHEMBL14940180 0.75 CYP2D6 (0.44) CYP2D6ALDH1A1TSHRMAPK1ALOX12
SCHEMBL14939045 0.71 CYP2D6 (0.42) CYP2D6ALDH1A1TSHRMAPK1ALOX12
SCHEMBL14939206 0.71 ALDH1A1 (0.45) CYP2D6ALDH1A1TSHRMAPK1ALOX12
SCHEMBL14940197 0.70 NPC1 (0.45) CYP2D6ALDH1A1TSHRMAPK1ALOX12
SCHEMBL14939120 0.70 CYP2D6 (0.45) CYP2D6ALDH1A1TSHRMAPK1ALOX12
SCHEMBL14939387 0.70 ALDH1A1 (0.45) CYP2D6ALDH1A1TSHRMAPK1ALOX12
SCHEMBL14939171 0.68 CYP2D6 (0.42) CYP2D6ALDH1A1TSHRMAPK1ALOX12
SCHEMBL14938972 0.67 CYP2D6 (0.41) CYP2D6ALDH1A1TSHRMAPK1ALOX12
SCHEMBL14939487 0.67 ALDH1A1 (0.45) CYP2D6ALDH1A1TSHRMAPK1ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed