SCHEMBL14939477

SCHEMBL14939477

O=C1c2ccccc2CC1(c1ccccc1)C1CCN(Cc2ccc3c(c2)OCO3)CC1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.53
NR1H4 Q96RI1 1/20 0.51
ALDH1A1 P00352 2/20 0.50
ALDH3A1 P30838 1/20 0.50
SIGMAR1 Q99720 2/20 0.49
TRPV6 Q9H1D0 1/20 0.48
LMNA P02545 2/20 0.48
KMT2A Q03164 4/20 0.47
MEN1 O00255 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HSD17B10 Q99714 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
MCHR1 Q99705 1/20 0.47
PKM P14618 1/20 0.47
FAAH O00519 1/20 0.46
DRD2 P14416 1/20 0.46
DRD4 P21917 1/20 0.46
CYP2D6 P10635 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940161 0.94 TSHR (0.49) TSHRNR1H4ALDH1A1ALDH3A1SIGMAR1
SCHEMBL14939192 0.91 ALDH1A1 (0.49) TSHRNR1H4ALDH1A1ALDH3A1SIGMAR1
SCHEMBL14939246 0.84 NPSR1 (0.53) SIGMAR1NPSR1DRD2
SCHEMBL14940051 0.84 NPSR1 (0.53) SIGMAR1NPSR1DRD2
SCHEMBL14939245 0.84 NPSR1 (0.53) SIGMAR1NPSR1DRD2
SCHEMBL14939923 0.83 CXCR3 (0.61) ALDH1A1SIGMAR1KMT2AMEN1NPSR1
SCHEMBL14939226 0.82 CXCR3 (0.61) SIGMAR1LMNANPSR1DRD2
SCHEMBL14939146 0.81 NR1H4 (0.53) TSHRNR1H4ALDH1A1ALDH3A1LMNA
SCHEMBL14939801 0.81 NR1H4 (0.53) TSHRNR1H4ALDH1A1ALDH3A1LMNA
SCHEMBL14939474 0.81 NR1H4 (0.53) TSHRNR1H4ALDH1A1ALDH3A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed