SCHEMBL14939480

SCHEMBL14939480

Cc1cccc(CN2CCN(C3(c4cccc(C)c4)Cc4ccccc4C3=O)CC2)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.48
CHRM2 P08172 3/20 0.45
CHRM3 P20309 3/20 0.45
ALDH1A1 P00352 6/20 0.44
KDM4E B2RXH2 4/20 0.44
HTT P42858 2/20 0.44
FAAH O00519 1/20 0.43
ACHE P22303 1/20 0.42
MAPT P10636 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
DRD2 P14416 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA9 Q16790 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939466 0.96 NPSR1 (0.54) NPSR1CHRM2CHRM3ALDH1A1KDM4E
SCHEMBL14939416 0.95 NPSR1 (0.45) NPSR1CHRM2CHRM3ALDH1A1KDM4E
SCHEMBL14939036 0.93 NPSR1 (0.47) NPSR1ALDH1A1KDM4EHTTMAPT
SCHEMBL14939908 0.91 SIGMAR1 (0.51) NPSR1CHRM2CHRM3ALDH1A1KDM4E
SCHEMBL14939643 0.90 ALDH1A1 (0.43) NPSR1CHRM2CHRM3ALDH1A1KDM4E
SCHEMBL14939534 0.88 ALDH1A1 (0.49) NPSR1ALDH1A1KDM4EHTTMAPT
SCHEMBL14939091 0.87 KMT2A (0.42) NPSR1ALDH1A1KDM4EHTTACHE
SCHEMBL14939559 0.87 KMT2A (0.42) NPSR1ALDH1A1KDM4EHTTACHE
SCHEMBL14939089 0.87 KMT2A (0.42) NPSR1ALDH1A1KDM4EHTTACHE
SCHEMBL14939007 0.87 NPSR1 (0.53) NPSR1ALDH1A1KDM4EHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed