SCHEMBL14939550

SCHEMBL14939550

Cc1cc(C2(Br)C(=O)c3ccccc3C2=O)ccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ2 O43526 1/20 0.44
CYP2D6 P10635 1/20 0.41
CDC7 O00311 1/20 0.40
ROCK2 O75116 1/20 0.40
MAP4K4 O95819 1/20 0.40
CDK2 P24941 1/20 0.40
GSK3B P49841 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
PDK2 Q15119 1/20 0.38
RECQL P46063 3/20 0.37
ALDH1A1 P00352 3/20 0.37
L3MBTL1 Q9Y468 3/20 0.37
BACE1 P56817 3/20 0.37
ALOX12 P18054 2/20 0.37
UHRF1 Q96T88 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939593 0.81 CYP2D6 (0.45) CYP2D6RECQLALDH1A1L3MBTL1BACE1
SCHEMBL14940158 0.76 NPSR1 (0.53) CYP2D6RECQLALDH1A1L3MBTL1BACE1
SCHEMBL14939588 0.75 ALDH1A1 (0.50) KCNQ2CYP2D6RECQLALDH1A1L3MBTL1
SCHEMBL14939045 0.75 CYP2D6 (0.42) KCNQ2CYP2D6RECQLALDH1A1L3MBTL1
SCHEMBL14939751 0.75 CYP2D6 (0.42) CYP2D6PDK2RECQLALDH1A1L3MBTL1
SCHEMBL14939640 0.75 KMT2A (0.41) CYP2D6RECQLALDH1A1L3MBTL1BACE1
SCHEMBL14940340 0.74 HRH4 (0.39) RECQLALDH1A1TSHRCASP1MAPT
SCHEMBL14939160 0.73 CYP2D6 (0.48) CYP2D6RECQLALDH1A1L3MBTL1BACE1
SCHEMBL14941913 0.73 CYP2D6 (0.38) CYP2D6RECQLALDH1A1L3MBTL1BACE1
SCHEMBL14939402 0.72 CYP2D6 (0.49) CYP2D6RECQLALDH1A1L3MBTL1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed