SCHEMBL14939633

SCHEMBL14939633

Cc1cc(F)cc(C2(N3CCN(Cc4ccc(C)cc4C)CC3)Cc3c(F)cccc3C2=O)c1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 3/20 0.36
GNRHR P30968 5/20 0.36
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
DRD2 P14416 1/20 0.35
DRD1 P21728 1/20 0.35
TDP1 Q9NUW8 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
COMT P21964 1/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939696 0.95 GRIN2B (0.38) GRIN2BGNRHRALDH1A1POLBL3MBTL1
SCHEMBL14939181 0.92 ALDH1A1 (0.41) GNRHRALDH1A1POLBL3MBTL1TDP1
SCHEMBL14940179 0.92 ALDH1A1 (0.37) GRIN2BGNRHRALDH1A1POLBL3MBTL1
SCHEMBL14939210 0.92 GRIN2B (0.38) GRIN2BGNRHRALDH1A1POLBL3MBTL1
SCHEMBL14938813 0.90 ALDH1A1 (0.36) ALDH1A1POLBSMN1; SMN2MAPTMAPK1
SCHEMBL14938749 0.89 ALDH1A1 (0.35) GNRHRALDH1A1L3MBTL1TDP1MAPT
SCHEMBL14939156 0.88 BCHE (0.35) ALDH1A1POLBMAPK1
SCHEMBL14940081 0.87 ALDH1A1 (0.44) ALDH1A1MAPT
SCHEMBL14938829 0.87 ALDH1A1 (0.41) GNRHRALDH1A1POLBL3MBTL1TDP1
SCHEMBL14939170 0.87 TP53 (0.39) GNRHRALDH1A1SMN1; SMN2MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed