SCHEMBL14939181

SCHEMBL14939181

Cc1cc(F)cc(C2(N3CCN(Cc4ccccc4C)CC3)Cc3c(F)cccc3C2=O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
GAA P10253 2/20 0.41
KDM4E B2RXH2 5/20 0.39
TDP1 Q9NUW8 2/20 0.39
KMT2A Q03164 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GNRHR P30968 1/20 0.36
CHRM1 P11229 2/20 0.36
MEN1 O00255 2/20 0.35
MAPK1 P28482 1/20 0.35
ATM Q13315 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CYP2A13 Q16696 1/20 0.34
ALDH3A1 P30838 1/20 0.34
RAB9A P51151 1/20 0.34
LMNA P02545 2/20 0.34
ACHE P22303 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14938829 0.95 ALDH1A1 (0.41) ALDH1A1GAAKDM4ETDP1KMT2A
SCHEMBL14938813 0.93 ALDH1A1 (0.36) ALDH1A1GAAKDM4EKMT2AMEN1
SCHEMBL14939633 0.92 GRIN2B (0.36) ALDH1A1TDP1L3MBTL1GNRHRMAPK1
SCHEMBL14938749 0.92 ALDH1A1 (0.35) ALDH1A1GAAKDM4ETDP1KMT2A
SCHEMBL14939170 0.91 TP53 (0.39) ALDH1A1GAAKDM4EKMT2AGNRHR
SCHEMBL14939125 0.91 ALDH1A1 (0.40) ALDH1A1GAAKDM4ETDP1KMT2A
SCHEMBL14939127 0.91 ALDH1A1 (0.40) ALDH1A1GAAKDM4ETDP1KMT2A
SCHEMBL14939319 0.91 ALDH1A1 (0.40) ALDH1A1GAAKDM4ETDP1KMT2A
SCHEMBL14940332 0.91 ALDH1A1 (0.47) ALDH1A1GAAKDM4ETDP1KMT2A
SCHEMBL14939156 0.89 BCHE (0.35) ALDH1A1GAAKDM4EKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed