SCHEMBL14939657

SCHEMBL14939657

CCc1ccccc1CN1CCN(C2(c3cccc(Br)n3)C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.46
ADORA2A P29274 5/20 0.36
ADORA1 P30542 5/20 0.36
CYP2D6 P10635 1/20 0.36
LMNA P02545 2/20 0.35
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
FAAH O00519 1/20 0.34
KMT2A Q03164 1/20 0.34
HTR7 P34969 1/20 0.34
TRPC5 Q9UL62 2/20 0.34
DPP8 Q6V1X1 1/20 0.34
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940304 0.90 NPSR1 (0.46) NPSR1LMNAKMT2ATRPC5MAPT
SCHEMBL14939217 0.88 NPSR1 (0.48) NPSR1FAAHKMT2AMAPT
SCHEMBL14939940 0.88 NPSR1 (0.47) NPSR1ADORA2AADORA1CYP2D6LMNA
SCHEMBL14939130 0.88 NPSR1 (0.47) NPSR1ADORA2AADORA1CYP2D6LMNA
SCHEMBL14940151 0.87 MEN1 (0.44) NPSR1CYP2D6DRD2KMT2AHTR7
SCHEMBL14939571 0.87 NPSR1 (0.49) NPSR1ADORA2AADORA1LMNAKMT2A
SCHEMBL14939341 0.85 NPSR1 (0.65) NPSR1LMNADRD2KMT2ATRPC5
SCHEMBL14939274 0.84 NPSR1 (0.44) NPSR1ADORA2AADORA1LMNADRD2
SCHEMBL14939260 0.83 NPSR1 (0.49) NPSR1CYP2D6LMNADRD2DRD3
SCHEMBL14940076 0.82 NPSR1 (0.46) NPSR1ADORA2AADORA1CYP2D6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed