SCHEMBL14939729

SCHEMBL14939729

Cc1cc(C2(N3CCN(Cc4ccccc4)CC3)C(=O)c3ccccc3C2=O)ccn1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.68
ADAM17 P78536 1/20 0.45
MAPT P10636 3/20 0.45
MMP2 P08253 2/20 0.43
MMP9 P14780 2/20 0.43
LMNA P02545 2/20 0.42
TSHR P16473 2/20 0.42
HTT P42858 1/20 0.42
POLB P06746 1/20 0.41
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
SIGMAR1 Q99720 3/20 0.40
DRD2 P14416 2/20 0.40
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
HTR2B P41595 2/20 0.40
NCF1 P14598 1/20 0.39
MC4R P32245 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939172 0.88 NPSR1 (0.53) NPSR1MAPTLMNATSHRALDH1A1
SCHEMBL14939533 0.87 NPSR1 (0.73) NPSR1ADAM17MAPTMMP2MMP9
SCHEMBL14939059 0.87 NPSR1 (0.51) NPSR1MAPTHTTALDH1A1GAA
SCHEMBL14939936 0.87 NPSR1 (0.50) NPSR1MAPTLMNAALDH1A1GAA
SCHEMBL14938836 0.87 NPSR1 (0.50) NPSR1ADAM17MAPTLMNA
SCHEMBL14939742 0.83 NPSR1 (0.82) NPSR1MAPTMMP2MMP9LMNA
SCHEMBL14940278 0.83 NPSR1 (0.67) NPSR1ADAM17MAPTMMP2MMP9
SCHEMBL14939733 0.83 NPSR1 (0.47) NPSR1MAPTTSHRHTTALDH1A1
SCHEMBL14939786 0.83 NPSR1 (0.62) NPSR1ADAM17MAPTMMP2MMP9
SCHEMBL14939558 0.83 NPSR1 (0.62) NPSR1ADAM17MAPTMMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed