SCHEMBL14939769

SCHEMBL14939769

O=C1c2ccccc2C(=O)C1(c1ccnc2ccccc12)N1CCN(Cc2ccccc2)CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.62
HTR1A P08908 1/20 0.46
HTR7 P34969 1/20 0.46
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 2/20 0.44
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
ADAM17 P78536 1/20 0.44
MAPT P10636 2/20 0.43
HPGD P15428 1/20 0.43
ACHE P22303 1/20 0.42
SIGMAR1 Q99720 3/20 0.41
TSHR P16473 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HIF1A Q16665 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
FAAH O00519 1/20 0.41
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
BCHE P06276 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940079 0.86 SIGMAR1 (0.50) NPSR1HTR1AALDH1A1KDM4EACHE
SCHEMBL14939310 0.86 NPSR1 (0.46) NPSR1ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL14939088 0.85 NPSR1 (0.46) NPSR1HTR1AALDH1A1KDM4ELMNA
SCHEMBL14939248 0.84 L3MBTL1 (0.53) HTR1AALDH1A1KDM4ESMN1; SMN2HPGD
SCHEMBL14939152 0.84 KDM4E (0.44) NPSR1HTR1AHTR7ALDH1A1KDM4E
SCHEMBL14938920 0.82 SIGMAR1 (0.43) NPSR1ALDH1A1KDM4ESIGMAR1MMP2
SCHEMBL14939412 0.80 NPSR1 (0.70) NPSR1HTR1ASIGMAR1MMP2MMP9
SCHEMBL14939887 0.78 NPSR1 (0.64) NPSR1ALDH1A1KDM4ELMNAADAM17
SCHEMBL14939617 0.78 NPSR1 (1.00) NPSR1LMNAMAPTSIGMAR1MMP2
SCHEMBL14939558 0.77 NPSR1 (0.62) NPSR1ALDH1A1LMNASMN1; SMN2ADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed