SCHEMBL14939852

SCHEMBL14939852

O=C1c2ccccc2CC1(c1cccc(F)c1)N1CCN(Cc2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.54
SIGMAR1 Q99720 7/20 0.46
DRD2 P14416 4/20 0.46
HTR2A P28223 4/20 0.46
HTR2C P28335 4/20 0.46
HTR2B P41595 4/20 0.46
ALDH1A1 P00352 2/20 0.44
ALDH3A1 P30838 1/20 0.44
CHRM2 P08172 1/20 0.43
CHRM3 P20309 1/20 0.43
OPRM1 P35372 1/20 0.43
KCNH2 Q12809 1/20 0.43
CYP2D6 P10635 1/20 0.42
MAPK1 P28482 1/20 0.42
FAAH O00519 1/20 0.41
MC4R P32245 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940002 0.96 NPSR1 (0.50) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14940059 0.94 NPSR1 (0.49) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14939844 0.92 NPSR1 (0.45) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14939129 0.90 NPSR1 (0.46) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14939625 0.89 NPSR1 (0.64) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14940373 0.89 NPSR1 (0.64) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14939175 0.89 NPSR1 (0.64) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14939219 0.89 NPSR1 (0.51) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14940465 0.88 SIGMAR1 (0.50) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939880 0.88 NPSR1 (0.52) NPSR1SIGMAR1DRD2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed