SCHEMBL14940230

SCHEMBL14940230

O=C1c2ccccc2C(=O)C1(c1cccc(Cl)c1)N1CCN(Cc2cc(F)ccc2F)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.55
MAPT P10636 3/20 0.45
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
DRD2 P14416 2/20 0.41
DRD1 P21728 1/20 0.41
HTR7 P34969 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
SIGMAR1 Q99720 2/20 0.37
ALDH3A1 P30838 1/20 0.36
RIPK1 Q13546 1/20 0.36
CHRM2 P08172 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940099 0.93 NPSR1 (0.55) NPSR1MAPTALDH1A1LMNAKMT2A
SCHEMBL14939168 0.91 MAPT (0.53) NPSR1MAPTALDH1A1LMNAKMT2A
SCHEMBL14939013 0.90 NPSR1 (0.64) NPSR1MAPTALDH1A1LMNAKMT2A
SCHEMBL14939616 0.89 NPSR1 (0.51) NPSR1MAPTALDH1A1LMNAKMT2A
SCHEMBL14939105 0.89 NPSR1 (0.51) NPSR1MAPTALDH1A1LMNAKMT2A
SCHEMBL14939492 0.87 NPSR1 (0.53) NPSR1MAPTALDH1A1LMNAKMT2A
SCHEMBL14939266 0.87 MAPT (0.55) NPSR1MAPTALDH1A1KDM4EDRD2
SCHEMBL14939874 0.86 NPSR1 (0.48) NPSR1MAPTALDH1A1LMNAKMT2A
SCHEMBL14939885 0.85 NPSR1 (0.59) NPSR1MAPTALDH1A1LMNAKMT2A
SCHEMBL14939155 0.84 NPSR1 (0.54) NPSR1MAPTALDH1A1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed