SCHEMBL14940320

SCHEMBL14940320

O=C1c2ccccc2C(=O)C1(c1cccc(C(F)(F)F)c1)N1CCN(Cc2ccccc2)CC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.72
MAPT P10636 1/20 0.64
OPRL1 P41146 3/20 0.50
CHRM3 P20309 1/20 0.48
LMNA P02545 3/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
GAA P10253 2/20 0.47
HTT P42858 2/20 0.47
KMT2A Q03164 1/20 0.47
CHRM4 P08173 1/20 0.47
TSHR P16473 1/20 0.47
FAAH O00519 1/20 0.47
SIGMAR1 Q99720 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
DRD4 P21917 1/20 0.45
TRPV6 Q9H1D0 1/20 0.45
TRPV5 Q9NQA5 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939093 0.87 MAPT (0.57) NPSR1MAPTOPRL1CHRM3KDM4E
SCHEMBL14940064 0.85 MAPT (0.52) NPSR1MAPTOPRL1LMNAKDM4E
SCHEMBL14939190 0.85 MAPT (0.57) NPSR1MAPTOPRL1LMNAKDM4E
SCHEMBL14939709 0.85 NPSR1 (0.77) NPSR1MAPTCHRM3LMNAALDH1A1
SCHEMBL14939617 0.84 NPSR1 (1.00) NPSR1MAPTLMNASIGMAR1
SCHEMBL14939425 0.84 NPSR1 (0.79) NPSR1MAPTCHRM3LMNAKDM4E
SCHEMBL14939266 0.83 MAPT (0.55) NPSR1MAPTOPRL1CHRM3KDM4E
SCHEMBL14939840 0.83 NPSR1 (0.77) NPSR1MAPTLMNAKDM4EKMT2A
SCHEMBL14939933 0.83 NPSR1 (0.77) NPSR1MAPTCHRM3LMNAKDM4E
SCHEMBL14940042 0.83 MAPT (0.54) NPSR1MAPTCHRM3LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed