SCHEMBL14940557

SCHEMBL14940557

NC(=O)C1=CNCc2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
NOTUM Q6P988 4/20 0.37
AURKA O14965 1/20 0.36
BCAT2 O15382 2/20 0.35
CYP3A4 P08684 2/20 0.34
MAPT P10636 2/20 0.34
BLM P54132 2/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 1/20 0.34
PABPC1 P11940 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 2/20 0.33
POLB P06746 1/20 0.33
PARP1 P09874 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2675467 0.84 CA12 (0.41) CA12CA9NOTUMMAPTKDM4E
SCHEMBL7385627 0.72 EGFR (0.35) CA12CA9NOTUMCYP3A4MAPT
SCHEMBL4527060 0.72 NOTUM (0.40) NOTUMBCAT2CYP3A4MAPTBLM
SCHEMBL4560301 0.69 IKBKB (0.47) CYP3A4MAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL8111658 0.69 NOTUM (0.45) NOTUMBCAT2MAPTKDM4EALDH1A1
SCHEMBL7391653 0.68 KEAP1 (0.43) CA12CA9NOTUMMAPTKDM4E
SCHEMBL21063661 0.68 MAOA (0.41) NOTUMBCAT2CYP3A4MAPTBLM
SCHEMBL28300619 0.68 CA12 (0.40) CA12CA9PARP1
SCHEMBL10783453 0.68 MAOA (0.44) NOTUMBCAT2CYP3A4MAPTBLM
SCHEMBL16247863 0.67 CA12 (0.42) CA12CA9ALDH1A1KMT2APARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023165591-A1 COMPOUNDS AND THEIR USES AS LPAR5 ANTAGONISTS IMMUTHER PHARMATECH (SHANGHAI) CO., LTD. (CN) 2023-09-07 WO claimed
EP-2780324-A1 HETEROCYCLIC CARBOXAMIDES USEFUL AS INHIBITORS OF PHOSPHODIESTERASE TYPE 10A Abbvie Deutschland GmbH & Co. KG (DE) 2014-09-24 EP claimed
WO-2013068489-A1 HETEROCYCLIC CARBOXAMIDES USEFUL AS INHIBITORS OF PHOSPHODIESTERASE TYPE 10A ABBOTT GMBH & CO. KG (DE) 2013-05-16 WO claimed
CN-116082232-A Monoamine oxidase inhibitor, preparation method and application thereof 浙江海洋大学 2023-05-09 CN disclosed
EP-3723753-A1 INHIBITORS OF FIBROBLAST ACTIVATION PROTEIN Praxis Biotech LLC (US) 2020-10-21 EP disclosed
WO-2019118932-A1 INHIBITORS OF FIBROBLAST ACTIVATION PROTEIN Praxis Biotech LLC (US) 2019-06-20 WO disclosed