SCHEMBL1494841

SCHEMBL1494841

NC(=O)C1CCN(c2cc(C(=O)O)ccn2)CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.62
TDP1 Q9NUW8 1/20 0.51
KDM4E B2RXH2 2/20 0.49
ABL1 P00519 1/20 0.49
LMNA P02545 1/20 0.49
KDM4C Q9H3R0 4/20 0.47
KDM4A O75164 2/20 0.47
PKM P14618 1/20 0.46
DPP4 P27487 1/20 0.46
TSHR P16473 1/20 0.46
KDM5A P29375 2/20 0.45
KDM5B Q9UGL1 2/20 0.45
ALDH1A1 P00352 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
RECQL P46063 1/20 0.45
ITGB2 P05107 2/20 0.45
ICAM1 P05362 2/20 0.45
ITGAL P20701 2/20 0.45
KMT2A Q03164 1/20 0.44
GABRP O00591 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16966428 0.86 PIK3CA (0.65) PIK3CAKDM4EKDM4CKDM4ADPP4
SCHEMBL3743262 0.84 PIK3CA (0.67) PIK3CAKDM4EKDM4CKDM4ADPP4
SCHEMBL25296404 0.83 PIK3CA (0.51) PIK3CATDP1KDM4ELMNANPSR1
SCHEMBL3738805 0.83 PIK3CA (0.65) PIK3CAKDM4EKDM4CKDM4ADPP4
SCHEMBL31143236 0.81 PIK3CA (0.74) PIK3CAKDM4EKDM4CKDM4AKDM5A
SCHEMBL1516867 0.81 PIK3CA (0.74) PIK3CAKDM4EKDM4CKDM4AKDM5A
SCHEMBL20950150 0.80 PIK3CA (0.60) PIK3CAKDM4CKDM4ADPP4KDM5A
SCHEMBL12552657 0.80 PIK3CA (0.60) PIK3CAKDM4CKDM4AKDM5AKDM5B
Hydrochloric Acid SCHEMBL1252523 0.79 PIK3CA (0.72) PIK3CAKDM4EKDM4CKDM4AKDM5A
SCHEMBL1255519 0.79 PIK3CA (0.72) PIK3CATDP1KDM4EKDM4CKDM4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110053915-A1 HETEROCYCLIC INHIBITORS OF AN Hh-SIGNAL CASCADE, MEDICINAL COMPOSITIONS BASED THEREON AND METHODS FOR TREATING DISEASES CAUSED BY THE ABERRANT ACTIVITY OF AN Hh-SIGNAL SYSTEM ALLA CHEM, LLC (US) 2011-03-03 US claimed
US-8486945-B2 Heterocyclic inhibitors of an Hh-signal cascade, medicinal compositions based thereon and methods for treating diseases caused by the aberrant activity of an Hh-signal system Ivachtchenko, Alexandre Vasilievich (US) 2013-07-16 US disclosed
US-20110053915-A1 HETEROCYCLIC INHIBITORS OF AN Hh-SIGNAL CASCADE, MEDICINAL COMPOSITIONS BASED THEREON AND METHODS FOR TREATING DISEASES CAUSED BY THE ABERRANT ACTIVITY OF AN Hh-SIGNAL SYSTEM ALLA CHEM, LLC (US) 2011-03-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110053915-A1 HETEROCYCLIC INHIBITORS OF AN Hh-SIGNAL CASCADE, MEDICINAL COMPOSITIONS BASED THEREON AND METHODS FOR TREATING DISEASES CAUSED BY THE ABERRANT ACTIVITY OF AN Hh-SIGNAL SYSTEM SHH, SMO, GLI1 PIK3CA 1145/4885TDP1 4579/4885KDM4E 2294/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.