SCHEMBL14950286

SCHEMBL14950286

Cc1cccc(-c2cn(C(=O)N(C)C3CCOCC3)cn2)c1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FAAH O00519 2/20 0.54
CES2 O00748 1/20 0.54
GRM5 P41594 2/20 0.40
GRIN2B Q13224 10/20 0.39
LMNA P02545 1/20 0.39
KMO O15229 2/20 0.37
TGFBR1 P36897 1/20 0.37
AVPR1B P47901 1/20 0.37
MCHR1 Q99705 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14950284 0.90 FAAH (0.66) FAAHCES2GRM5GRIN2BKMO
SCHEMBL427868 0.90 FAAH (0.59) FAAHCES2TGFBR1
SCHEMBL526192 0.89 FAAH (0.67) FAAHCES2GRM5KMO
SCHEMBL14950261 0.89 FAAH (0.53) FAAHCES2GRIN2BLMNATGFBR1
SCHEMBL16424253 0.88 FAAH (0.53) FAAHCES2TGFBR1
SCHEMBL427343 0.85 FAAH (0.54) FAAHCES2TGFBR1
SCHEMBL14937765 0.85 FAAH (0.52) FAAHCES2LMNA
SCHEMBL14950257 0.84 FAAH (0.52) FAAHCES2GRIN2B
SCHEMBL427732 0.84 FAAH (0.53) FAAHCES2TGFBR1MCHR1
SCHEMBL426220 0.84 FAAH (0.53) FAAHCES2TGFBR1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130123493-A1 PROCESS FOR THE SYNTHESIS OF SUBSTITUTED UREA COMPOUNDS BIAL - PORTELA & CA, S.A. (PT) 2013-05-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130123493-A1 PROCESS FOR THE SYNTHESIS OF SUBSTITUTED UREA COMPOUNDS UTS2R, ARG1, PRMT1 FAAH 2166/4885CES2 463/4885GRM5 3634/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.