SCHEMBL14950656

SCHEMBL14950656

Oc1ccc(SC(c2ccccc2)(c2ccccc2)c2ccccc2)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.41
KIF11 P52732 8/20 0.40
ESR1 P03372 8/20 0.36
ESR2 Q92731 5/20 0.36
TTR P02766 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14937782 0.79 LDHA (0.41) KIF11ALDH1A1
SCHEMBL14950659 0.77 KIF11 (0.38) KIF11ESR1ESR2ALDH1A1CYP3A4
SCHEMBL28229893 0.74 HSD17B10 (0.46) HSD17B10ESR1ESR2TTRCYP3A4
SCHEMBL67991 0.71 HSD17B10 (0.56) HSD17B10ESR1ESR2TTRALDH1A1
SCHEMBL30821022 0.70 KIF11 (0.38) HSD17B10KIF11ESR1ESR2ALDH1A1
SCHEMBL5307183 0.69 KIF11 (0.50) HSD17B10KIF11ESR1ESR2ALDH1A1
SCHEMBL14937828 0.68 PPARG (0.37) KIF11
SCHEMBL5878646 0.67 HSD17B10 (0.52) HSD17B10ESR1ESR2TTRCYP3A4
SCHEMBL19691959 0.66 POLB (0.44) HSD17B10KIF11ALDH1A1
SCHEMBL28736885 0.66 TSHR (0.34) KIF11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2776392-B1 PROCESS FOR THE PREPARATION OF 1-ACYL-4-PHENYLSULFONYLPROLINAMIDE DERIVATIVES AND NEW INTERMEDIATES HOFFMANN LA ROCHE (CH) 2016-05-18 EP disclosed
WO-2013068434-A1 PROCESS FOR THE PREPARATION OF 1-ACYL-4-PHENYLSULFONYLPROLINAMIDE DERIVATIVES AND NEW INTERMEDIATES F. HOFFMANN-LA ROCHE AG (CH) 2013-05-16 WO disclosed