SCHEMBL149537

SCHEMBL149537

Clc1ncc2ccccc2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
EGFR P00533 2/20 0.46
GPR3 P46089 1/20 0.46
ALDH1A1 P00352 3/20 0.44
MAPT P10636 2/20 0.44
GLA P06280 1/20 0.44
HPGD P15428 1/20 0.44
ACHE P22303 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
CYP1A2 P05177 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
HTR3A P46098 1/20 0.42
HRH4 Q9H3N8 1/20 0.42
KMT2A Q03164 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 1/20 0.38
NCF1 P14598 1/20 0.38
NOS2 P35228 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29666411 1.00 KDM4E (0.46) KDM4EEGFRGPR3ALDH1A1MAPT
SCHEMBL30100747 1.00 KDM4E (0.46) KDM4EEGFRGPR3ALDH1A1MAPT
Hydrochloric Acid SCHEMBL10524097 0.98 KDM4E (0.45) KDM4EEGFRGPR3ALDH1A1MAPT
Formaldehyde SCHEMBL27640099 0.94 KDM4E (0.42) KDM4EEGFRGPR3ALDH1A1MAPT
Biphenyl SCHEMBL28365892 0.92 NPC1 (0.44) KDM4EEGFRGPR3ALDH1A1GLA
SCHEMBL20163588 0.88 EGFR (0.38) KDM4EEGFRGPR3ALDH1A1MAPT
SCHEMBL29520469 0.80 CYP1A2 (0.44) KDM4EEGFRGPR3ALDH1A1MAPT
Valine SCHEMBL9998032 0.76 SLC7A5 (0.42) KDM4EALDH1A1CYP1A2SMN1; SMN2RAB9A
SCHEMBL30198446 0.75 CYP1A2 (0.60) KDM4EEGFRGPR3ALDH1A1MAPT
SCHEMBL30527184 0.75 CYP1A2 (0.60) KDM4EEGFRGPR3ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1262 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117486809-A 2-chloroquinazoline compound, preparation method and application thereof in preparation of medicines for preventing or treating breast cancer 浙江工业大学 2024-02-02 CN claimed
CN-114920704-B Phenyl piperazine quinazoline compound or pharmaceutically acceptable salt thereof, preparation method and application 暨南大学 2023-11-03 CN claimed
CN-114886896-B Application of 2-chloroquinazoline derivative or pharmaceutically acceptable salt thereof in preparation of medicines for preventing or treating cervical cancer 浙江工业大学 2023-07-14 CN claimed
CN-114920704-A Phenyl piperazine quinazoline compound or pharmaceutically acceptable salt thereof, preparation method and application 暨南大学 2022-08-19 CN claimed
CN-114886896-A Application of 2-chloroquinazoline derivative or pharmaceutically acceptable salt thereof in preparation of drugs for preventing or treating cervical cancer 浙江工业大学 2022-08-12 CN claimed
CN-112300082-B Phenyl piperazine quinazoline compound or pharmaceutically acceptable salt thereof, preparation method and application 暨南大学 2022-04-26 CN claimed
WO-2021017996-A1 PHENYLPIPERAZINE QUINAZOLINE COMPOUND OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, AND PREPARATION METHOD THEREFOR AND USE THEREOF 暨南大学 2021-02-04 WO claimed
CN-112300082-A Phenyl piperazine quinazoline compound or pharmaceutically acceptable salt thereof, preparation method and application 暨南大学 2021-02-02 CN claimed
CN-105520951-B The polysaccharid derivative of toroidal shell containing quinazoline and preparation method and bioactivity 鲁东大学 2018-09-18 CN claimed
CN-104230826-B 2 fluoro quinazoline cyclics and preparation method thereof and pharmaceutical usage 复旦大学 2017-03-29 CN claimed
US-20150141421-A1 6,7-DIALKOXY QUINAZOLINE DERIVATIVES AND METHODS OF TREATING DRUG RESISTANT AND OTHER TUMORS NATCO PHARMA LIMITED (IN) 2015-05-21 US claimed
CN-102702178-B Process for the preparation of lapatinib and the salts thereof ITALIANA SINT SPA 2015-03-04 CN claimed
US-20110034459-A1 6,7-DIALKOXY QUINAZOLINE DERIVATIVES AND METHODS OF TREATING DRUG RESISTANT AND OTHER TUMORS NATCO PHARMA LTD. (IN) 2011-02-10 US claimed
EP-0954315-A2 USE OF QUINAZOLINE DERIVATIVES FOR THE MANUFACTURE OF A MEDICAMENT IN THE TREATMENT OF HYPERPROLIFERATIVE SKIN DISORDERS Sugen, Inc. (US) 1999-11-10 EP claimed
WO-1998010767-A9 USE OF QUINAZOLINE DERIVATIVES FOR THE MANUFACTURE OF A MEDICAMENT IN THE TREATMENT OF HYPERPROLIFERATIVE SKIN DISORDERS 1998-07-02 WO claimed
WO-1998010767-A2 USE OF QUINAZOLINE DERIVATIVES FOR THE MANUFACTURE OF A MEDICAMENT IN THE TREATMENT OF HYPERPROLIFERATIVE SKIN DISORDERS SUGEN, INC. (US) 1998-03-19 WO claimed
CN-121248582-B CDK12/PARP double-target inhibitor and preparation method and application thereof SOUTH CHINA UNIVERSITY OF TECHNOLOGY (CN) 2026-05-26 CN disclosed
US-20260137684-A1 ROCK2 Inhibitors And Uses Thereof RESTOR PHARMACEUTICALS (US) 2026-05-21 US disclosed
US-4133955-A Process for the production of 2-equivalent yellow couplers AGFA-GEVAERT AKTIENGESELLSCHAFT (DE) 1979-01-09 US disclosed
US-4098788-A Process for preparing quinazolines BRISTOL-MYERS COMPANY (US) 1978-07-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110034459-A1 6,7-DIALKOXY QUINAZOLINE DERIVATIVES AND METHODS OF TREATING DRUG RESISTANT AND OTHER TUMORS ERBB2, EGFR, ERBB3 KDM4E 2923/4885EGFR 2/4885GPR3 156/4885
US-20150141421-A1 6,7-DIALKOXY QUINAZOLINE DERIVATIVES AND METHODS OF TREATING DRUG RESISTANT AND OTHER TUMORS ERBB2, EGFR, GRK3 KDM4E 3005/4885EGFR 2/4885GPR3 92/4885
US-20260137684-A1 ROCK2 Inhibitors And Uses Thereof ROCK2, ROCK1, RHOA KDM4E 1974/4885EGFR 1956/4885GPR3 1678/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.