SCHEMBL14959151

SCHEMBL14959151

CN(C)C(=O)Cc1ccc(F)cc1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.62
POLB P06746 1/20 0.62
APEX1 P27695 1/20 0.62
SMN1; SMN2 Q16637 2/20 0.56
GAA P10253 2/20 0.48
CTBP2 P56545 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
LMNA P02545 1/20 0.46
KMT2A Q03164 1/20 0.46
HTT P42858 1/20 0.46
KDM4E B2RXH2 1/20 0.46
GABRA1 P14867 1/20 0.46
GABRB2 P47870 1/20 0.46
ALDH1A1 P00352 1/20 0.45
MAPK1 P28482 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6625005 0.84 TDP1 (0.59) TDP1POLBAPEX1SMN1; SMN2GAA
SCHEMBL14415483 0.82 TDP1 (0.62) TDP1POLBAPEX1SMN1; SMN2GAA
SCHEMBL1399311 0.81 TDP1 (0.56) TDP1POLBAPEX1SMN1; SMN2GAA
SCHEMBL4462525 0.81 TDP1 (0.56) TDP1POLBAPEX1SMN1; SMN2GAA
SCHEMBL14340565 0.81 ALDH1A1 (0.48) TDP1POLBAPEX1SMN1; SMN2HDAC4
SCHEMBL15920608 0.81 HDAC4 (0.44) TDP1POLBAPEX1HDAC4HDAC6
SCHEMBL10567198 0.81 CA2 (0.56) TDP1POLBAPEX1GAALMNA
SCHEMBL171877 0.81 CTBP2 (0.48) TDP1POLBAPEX1CTBP2HDAC4
SCHEMBL1973647 0.81 CA2 (0.56) CTBP2HDAC4HDAC6LMNA
SCHEMBL20888575 0.81 CA12 (0.56) TDP1POLBAPEX1SMN1; SMN2HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8445473-B2 Heteroaryl-substituted bicyclic Smac mimetics and the uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2013-05-21 US disclosed