SCHEMBL1495987

SCHEMBL1495987

Cn1ncc2c1Nc1cc(Cl)ccc1N(C(=O)C1CCC(CNC(=O)C3CCN(CCC(C)(C)C)CC3)CC1)C2

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CACNA1I Q9P0X4 9/20 0.43
KCNH2 Q12809 6/20 0.43
IDH1 O75874 4/20 0.37
AVPR1A P37288 7/20 0.37
OXTR P30559 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1496255 0.91 IDH1 (0.38) IDH1AVPR1AOXTR
SCHEMBL1495930 0.91 AVPR1A (0.40) IDH1AVPR1AOXTR
SCHEMBL1496011 0.91 AVPR1A (0.41) CACNA1IKCNH2AVPR1AOXTR
SCHEMBL1495887 0.90 AVPR1A (0.45) IDH1AVPR1AOXTR
SCHEMBL1495936 0.84 DRD2 (0.41) IDH1AVPR1AOXTR
SCHEMBL2629001 0.83 IDH1 (0.37) IDH1AVPR1AOXTR
SCHEMBL2628459 0.83 IDH1 (0.40) IDH1AVPR1AOXTR
SCHEMBL1496052 0.83 AVPR1A (0.39) IDH1AVPR1AOXTR
SCHEMBL1496024 0.83 AVPR1A (0.43) CACNA1IAVPR1AOXTR
SCHEMBL2131177 0.83 AVPR1A (0.44) AVPR1AOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2292621-A1 Vasopressin v1a antagonists Vantia Limited (GB) 2011-03-09 EP claimed