SCHEMBL14960376

SCHEMBL14960376

CC(=O)c1ccc(-c2cc(C(F)(F)F)n(CF)n2)s1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
GAA P10253 3/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40
GABRA2 P47869 1/20 0.40
GABRB2 P47870 1/20 0.40
GABRA4 P48169 1/20 0.40
GABRE P78334 1/20 0.40
GABRA6 Q16445 1/20 0.40
GABRG1 Q8N1C3 1/20 0.40
GABRG3 Q99928 1/20 0.40
GABRQ Q9UN88 1/20 0.40
HDAC6 Q9UBN7 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14960293 0.91 ALDH1A1 (0.46) ALDH1A1GAAL3MBTL1GABRPGABRD
SCHEMBL1574357 0.83 ALDH1A1 (0.74) ALDH1A1GAAL3MBTL1GABRPGABRD
SCHEMBL14412375 0.81 ALDH1A1 (0.53) ALDH1A1GAAL3MBTL1HDAC6HDAC3
SCHEMBL14412177 0.80 NPC1 (0.50) ALDH1A1HDAC6HDAC3HDAC4HDAC1
SCHEMBL5212779 0.80 ALDH1A1 (0.53) ALDH1A1GAAL3MBTL1HDAC6HDAC3
SCHEMBL14412199 0.79 ALDH1A1 (0.51) ALDH1A1GAAHDAC6HDAC3HDAC4
SCHEMBL14412418 0.79 ALDH1A1 (0.50) ALDH1A1GAAL3MBTL1RAB9ANPC1
SCHEMBL14412372 0.78 ALDH1A1 (0.42) ALDH1A1HDAC6HDAC3HDAC4HDAC1
SCHEMBL14412392 0.77 ALDH1A1 (0.41) ALDH1A1GAAHDAC4CYP2C9MAPT
SCHEMBL14412290 0.77 ALDH1A1 (0.39) ALDH1A1GAAL3MBTL1LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1989185-B1 THERAPEUTIC COMPOUNDS HELICON THERAPEUTICS INC (US) 2013-05-22 EP disclosed