SCHEMBL14964774

SCHEMBL14964774

c1ccc(-c2csc3ncnc(N4CCC(CNCC5CC5)CC4)c23)cc1

nearest known ligand 0.83

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.66
HTT P42858 1/20 0.66
KMT2A Q03164 1/20 0.66
LMNA P02545 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16293150 0.93 POLB (0.61) POLBHTTKMT2ALMNA
SCHEMBL14965176 0.90 POLB (0.60) POLBHTTKMT2ALMNA
SCHEMBL14965126 0.90 ADRB2 (0.60) POLBHTTKMT2A
SCHEMBL17599008 0.90 KMT2A (0.77) POLBHTTKMT2ALMNA
SCHEMBL16293434 0.89 ADRB2 (0.64) LMNA
SCHEMBL27978763 0.89 STAT3 (0.59) POLBHTTKMT2ALMNA
SCHEMBL14965145 0.89 POLB (0.61) POLBHTTKMT2A
SCHEMBL14965467 0.88 POLB (0.60) POLBHTTKMT2A
SCHEMBL14965361 0.88 POLB (0.62) POLBHTTKMT2A
SCHEMBL14965357 0.88 ADRB2 (0.62) POLBHTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780343-A1 THIENO- AND FURO - PYRIMIDINES AND PYRIDINES, USEFUL AS POTASSIUM CHANNEL INHIBITORS Xention Limited (GB) 2014-09-24 EP disclosed
CN-104011054-A Thieno- and furo-pyrimidines and pyridines, useful as potassium channel inhibitors XENTION LTD 2014-08-27 CN disclosed
WO-2013072694-A1 THIENO- AND FURO - PYRIMIDINES AND PYRIDINES, USEFUL AS POTASSIUM CHANNEL INHIBITORS XENTION LIMITED (GB) 2013-05-23 WO disclosed