SCHEMBL14965286

SCHEMBL14965286

N#Cc1sc2nccc(N3CCC(COCCN4CCCC4)CC3)c2c1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14964972 0.90 HRH3 (0.39) CDK8
SCHEMBL14969446 0.86 MEN1 (0.45)
SCHEMBL14964799 0.81 KDM4E (0.37) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL14965154 0.80
SCHEMBL14968820 0.79 KDM4E (0.37) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL14964787 0.77 KDM4E (0.33) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL16293967 0.76
SCHEMBL16293417 0.74
SCHEMBL28087471 0.73 LTA4H (0.40) KDM4E
SCHEMBL14965203 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780343-A1 THIENO- AND FURO - PYRIMIDINES AND PYRIDINES, USEFUL AS POTASSIUM CHANNEL INHIBITORS Xention Limited (GB) 2014-09-24 EP disclosed
CN-104011054-A Thieno- and furo-pyrimidines and pyridines, useful as potassium channel inhibitors XENTION LTD 2014-08-27 CN disclosed
WO-2013072694-A1 THIENO- AND FURO - PYRIMIDINES AND PYRIDINES, USEFUL AS POTASSIUM CHANNEL INHIBITORS XENTION LIMITED (GB) 2013-05-23 WO disclosed