SCHEMBL14965621

SCHEMBL14965621

O=C(c1cccc(OC(F)(F)F)c1)N1CC(CN2CCOc3nc([N+](=O)[O-])cn3CC2)C1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.44
PDE2A O00408 2/20 0.41
KCNH2 Q12809 4/20 0.41
HSD11B1 P28845 1/20 0.39
MGLL Q99685 3/20 0.39
RAB9A P51151 1/20 0.38
KCNK3 O14649 2/20 0.38
KCNK9 Q9NPC2 2/20 0.38
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
CACNA1B Q00975 1/20 0.35
MAPK7 Q13164 1/20 0.35
ABL1 P00519 1/20 0.35
PTGS1 P23219 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966212 0.93 HSD11B1 (0.44) CHRM1PDE2AKCNH2HSD11B1MGLL
SCHEMBL14965524 0.91 CHRM1 (0.51) CHRM1KCNH2HSD11B1MGLLMAPK7
SCHEMBL14965843 0.84 CHRM1 (0.48) CHRM1KCNH2HSD11B1MGLLMAPK7
SCHEMBL14965637 0.82 CHRM1 (0.51) CHRM1KCNH2PTGS1SLC6A2SLC6A4
SCHEMBL14965784 0.80 CHRM1 (0.49) CHRM1KCNH2MGLLALDH1A1KDM4E
SCHEMBL14965916 0.79 ABL1 (0.56) CHRM1KCNH2RAB9AALDH1A1ABL1
SCHEMBL14966146 0.78 CHRM1 (0.36) CHRM1KCNH2ALDH1A1
SCHEMBL14965557 0.78 DRD4 (0.48) CHRM1KCNH2ALDH1A1
SCHEMBL14965586 0.77 EPHX2 (0.51) CHRM1KCNH2MAPT
SCHEMBL14965849 0.77 CHRM1 (0.44) CHRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed