SCHEMBL14965849

SCHEMBL14965849

O=C(CN1CCOc2nc([N+](=O)[O-])cn2CC1)NCc1cccc(OC(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.44
KCNH2 Q12809 4/20 0.43
GLS O94925 4/20 0.39
EPHX2 P34913 1/20 0.39
PTGER1 P34995 1/20 0.39
USP2 O75604 1/20 0.39
HTT P42858 1/20 0.39
GFER P55789 1/20 0.39
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
MAPK14 Q16539 1/20 0.38
POLB P06746 1/20 0.38
CHRM3 P20309 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965929 0.91 USP2 (0.39) USP2HTTGFERROCK2ROCK1
SCHEMBL14965548 0.90 CHRM1 (0.52) CHRM1KCNH2USP2HTT
SCHEMBL14965622 0.88 CHRM1 (0.50) CHRM1KCNH2USP2HTT
SCHEMBL14966262 0.88 POLB (0.49) USP2HTTPOLB
SCHEMBL14965557 0.87 DRD4 (0.48) CHRM1KCNH2EPHX2
SCHEMBL14965591 0.87 CHRM3 (0.47) CHRM1KCNH2ROCK2ROCK1MAPK14
SCHEMBL14965784 0.86 CHRM1 (0.49) CHRM1KCNH2HTTROCK2ROCK1
SCHEMBL14966200 0.86 CHRM1 (0.44) CHRM1KCNH2EPHX2
SCHEMBL14966219 0.83 CA1 (0.48) CHRM1KCNH2USP2HTTPOLB
SCHEMBL14965804 0.82 KMT2A (0.41) CHRM1KCNH2USP2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed