SCHEMBL14965644

SCHEMBL14965644

O=C(CN1CCOc2nc([N+](=O)[O-])cn2CC1)Nc1ccc(C(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA7 P43166 1/20 0.46
CACNA1G O43497 1/20 0.46
CACNA1B Q00975 1/20 0.46
KCNH2 Q12809 1/20 0.46
LMNA P02545 2/20 0.43
ATM Q13315 1/20 0.42
KMT2A Q03164 1/20 0.41
POLB P06746 3/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
IDO1 P14902 1/20 0.40
TDO2 P48775 1/20 0.40
CA9 Q16790 1/20 0.39
HIF1A Q16665 1/20 0.39
EPAS1 Q99814 1/20 0.39
CETP P11597 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966114 0.91 KCNH2 (0.38) CA1CA2CA7CACNA1GCACNA1B
SCHEMBL14966065 0.90 LMNA (0.54) LMNAKMT2APOLBL3MBTL1ALDH1A1
SCHEMBL14966219 0.88 CA1 (0.48) CA1CA2CA7KCNH2KMT2A
SCHEMBL14965783 0.86 NPC1 (0.51) LMNAATMKMT2APOLBALDH1A1
SCHEMBL14965587 0.85 HIF1A (0.60) KMT2AHIF1AEPAS1ALDH1A1
SCHEMBL14966242 0.83 LMNA (0.44) LMNAKMT2APOLBL3MBTL1ALDH1A1
SCHEMBL14965557 0.82 DRD4 (0.48) KCNH2ATMKMT2AALDH1A1
SCHEMBL14965837 0.82 HIF1A (0.44) KCNH2LMNAL3MBTL1HIF1AEPAS1
SCHEMBL14966262 0.81 POLB (0.49) LMNAKMT2APOLBL3MBTL1ALDH1A1
SCHEMBL5542906 0.81 KCNH2 (0.50) CA1CA2CA7CACNA1GCACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed