SCHEMBL14966262

SCHEMBL14966262

O=C(CN1CCOc2nc([N+](=O)[O-])cn2CC1)NCc1cccc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.49
ALDH1A1 P00352 3/20 0.43
CCR1 P32246 1/20 0.41
ATG4B Q9Y4P1 1/20 0.41
USP2 O75604 1/20 0.40
HTT P42858 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MAPT P10636 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966331 0.92 LMNA (0.45) POLBALDH1A1CCR1MAPTKMT2A
SCHEMBL14966219 0.90 CA1 (0.48) POLBALDH1A1ATG4BUSP2HTT
SCHEMBL14965849 0.88 CHRM1 (0.44) POLBUSP2HTT
SCHEMBL14966065 0.87 LMNA (0.54) POLBALDH1A1MAPTL3MBTL1TSHR
SCHEMBL14965929 0.85 USP2 (0.39) POLBALDH1A1USP2HTTKMT2A
SCHEMBL14966242 0.85 LMNA (0.44) POLBALDH1A1MAPTL3MBTL1TSHR
SCHEMBL14965968 0.85 LMNA (0.48) ALDH1A1LMNA
SCHEMBL14965548 0.83 CHRM1 (0.52) USP2HTTKMT2A
SCHEMBL14965565 0.82 KMT2A (0.43) ALDH1A1USP2HTTMAPTL3MBTL1
SCHEMBL14965644 0.81 CA1 (0.46) POLBALDH1A1HTTL3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed