SCHEMBL14965647

SCHEMBL14965647

CN1CCN(C(=O)c2cc(-c3cccc(CN4CCOc5nc([N+](=O)[O-])cn5CC4)n3)ccc2F)CC1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIK3R1 P27986 2/20 0.35
PIK3CA P42336 2/20 0.35
JAK2 O60674 3/20 0.35
JAK1 P23458 3/20 0.35
TYK2 P29597 3/20 0.35
JAK3 P52333 3/20 0.35
PARP1 P09874 2/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
ALDH1A1 P00352 4/20 0.34
HTT P42858 3/20 0.34
KDM4E B2RXH2 2/20 0.34
KCNK3 O14649 1/20 0.34
KCNK9 Q9NPC2 1/20 0.34
LMNA P02545 2/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966153 0.94 JAK2 (0.38) PIK3R1PIK3CAJAK2JAK1TYK2
SCHEMBL14966064 0.94 JAK2 (0.34) PIK3R1PIK3CAJAK2JAK1TYK2
SCHEMBL14966353 0.88 JAK2 (0.37) JAK2JAK1TYK2JAK3SMN1; SMN2
SCHEMBL14966011 0.88 MTOR (0.37) PIK3R1PIK3CAJAK2JAK1TYK2
SCHEMBL14966144 0.86 JAK2 (0.38) JAK2JAK1TYK2JAK3PARP1
SCHEMBL14965956 0.86 MTOR (0.39)
SCHEMBL14965639 0.86 AVPR1B (0.34)
SCHEMBL14966086 0.84 FGFR1 (0.38) ALDH1A1
SCHEMBL14965570 0.83 JAK2 (0.36) PIK3R1PIK3CAJAK2JAK1TYK2
SCHEMBL14965762 0.82 MTOR (0.39) JAK2JAK1TYK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed