SCHEMBL14965639

SCHEMBL14965639

CC(C)NC(=O)c1cc(-c2cccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)n2)ccc1F

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 8/20 0.34
SRC P12931 1/20 0.32
SCN9A Q15858 1/20 0.32
BACE1 P56817 1/20 0.32
MAPT P10636 1/20 0.31
KCNH2 Q12809 3/20 0.31
HTR1A P08908 1/20 0.31
DRD2 P14416 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
CHRM3 P20309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966213 0.94 HDAC4 (0.37) AVPR1BSRCSCN9AKCNH2
SCHEMBL14965956 0.91 MTOR (0.39) KCNH2HTR1ADRD2CHRM3
SCHEMBL14966086 0.89 FGFR1 (0.38) BACE1
SCHEMBL14966064 0.88 JAK2 (0.34) HTR1ADRD2
SCHEMBL14966011 0.88 MTOR (0.37) SRCSCN9AKCNH2HTR1ADRD2
SCHEMBL14965848 0.88 MCHR1 (0.37) AVPR1BKCNH2
SCHEMBL14966157 0.86 AVPR1B (0.38) AVPR1B
SCHEMBL14965647 0.86 PIK3R1 (0.35)
SCHEMBL14965762 0.85 MTOR (0.39) KCNH2CHRM3
SCHEMBL14966353 0.83 JAK2 (0.37) KCNH2HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed