SCHEMBL14965762

SCHEMBL14965762

CCNC(=O)c1ccc(-c2cccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)n2)cc1F

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.39
MAPK1 P28482 3/20 0.34
MET P08581 3/20 0.34
CHRM3 P20309 1/20 0.33
CHRM4 P08173 1/20 0.33
JAK2 O60674 2/20 0.32
JAK1 P23458 1/20 0.32
TYK2 P29597 1/20 0.32
JAK3 P52333 1/20 0.32
KCNH2 Q12809 1/20 0.32
MOK Q9UQ07 1/20 0.32
ACP1 P24666 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965956 0.94 MTOR (0.39) MTORCHRM3KCNH2HSP90AA1HSP90AB1
SCHEMBL14966213 0.91 HDAC4 (0.37) MAPK1METJAK2JAK1TYK2
SCHEMBL14965831 0.89 FGFR1 (0.36) MAPK1MET
SCHEMBL14965570 0.88 JAK2 (0.36) MTORMETJAK2JAK1TYK2
SCHEMBL14966353 0.87 JAK2 (0.37) METJAK2JAK1TYK2JAK3
SCHEMBL14966153 0.86 JAK2 (0.38) MTORMETJAK2JAK1TYK2
SCHEMBL14965597 0.86 MTOR (0.39) MTORMAPK1METCHRM4KCNH2
SCHEMBL14966211 0.86 MTOR (0.38) MTORMETCHRM4KCNH2HSP90AA1
SCHEMBL14965639 0.85 AVPR1B (0.34) CHRM3KCNH2
SCHEMBL14966011 0.84 MTOR (0.37) MTORJAK2JAK1TYK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed