SCHEMBL14965722

SCHEMBL14965722

O=C(NCc1cccc(F)c1)c1ccc(CN2CCOc3nc([N+](=O)[O-])cn3CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 3/20 0.48
KLK1 P06870 3/20 0.48
ALDH1A1 P00352 4/20 0.46
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CHRM3 P20309 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
TP53 P04637 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
HTR2C P28335 1/20 0.41
MCHR1 Q99705 1/20 0.41
HDAC4 P56524 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
ROCK2 O75116 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965800 0.90 ALDH1A1 (0.58) KLKB1KLK1ALDH1A1MEN1KMT2A
SCHEMBL14966210 0.89 ALDH1A1 (0.43) KLKB1KLK1ALDH1A1MEN1KMT2A
SCHEMBL14966045 0.88 TSHR (0.50) KLKB1KLK1ALDH1A1MEN1KMT2A
SCHEMBL14965591 0.88 CHRM3 (0.47) KLKB1KLK1ALDH1A1MEN1KMT2A
SCHEMBL14965538 0.86 HDAC4 (0.49) ALDH1A1CHRM3SMN1; SMN2HDAC4HDAC6
SCHEMBL14966186 0.86 ALDH1A1 (0.48) ALDH1A1MEN1KMT2ASMN1; SMN2NPC1
SCHEMBL14965370 0.84 ALDH1A1 (0.44) ALDH1A1MEN1KMT2ASMN1; SMN2NPC1
SCHEMBL14965856 0.84 PRKAA2 (0.46) ALDH1A1CHRM3SMN1; SMN2HDAC4HDAC6
SCHEMBL14965611 0.84 TSHR (0.61) KLKB1KLK1ALDH1A1MEN1KMT2A
SCHEMBL14965754 0.83 TSHR (0.47) ALDH1A1MEN1KMT2ASMN1; SMN2HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed