SCHEMBL14965800

SCHEMBL14965800

O=C(NCc1ccccc1)c1ccc(CN2CCOc3nc([N+](=O)[O-])cn3CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.58
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
TSHR P16473 1/20 0.46
MLLT1 Q03111 1/20 0.44
HDAC4 P56524 2/20 0.44
PRKAA2 P54646 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
KCNH2 Q12809 1/20 0.44
HDAC1 Q13547 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
MCHR1 Q99705 1/20 0.43
KLKB1 P03952 1/20 0.43
KLK1 P06870 1/20 0.43
HIF1A Q16665 1/20 0.42
EPAS1 Q99814 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966186 0.92 ALDH1A1 (0.48) ALDH1A1MEN1KMT2ATSHRMLLT1
SCHEMBL14965538 0.91 HDAC4 (0.49) ALDH1A1TSHRMLLT1HDAC4SMN1; SMN2
SCHEMBL14965722 0.90 KLKB1 (0.48) ALDH1A1MEN1KMT2ATSHRHDAC4
SCHEMBL14965856 0.90 PRKAA2 (0.46) ALDH1A1TSHRMLLT1HDAC4PRKAA2
SCHEMBL14965611 0.90 TSHR (0.61) ALDH1A1MEN1KMT2ATSHRMLLT1
SCHEMBL14965777 0.89 HIF1A (0.58) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL14965370 0.88 ALDH1A1 (0.44) ALDH1A1MEN1KMT2ATSHRMLLT1
SCHEMBL14966045 0.88 TSHR (0.50) ALDH1A1MEN1KMT2ATSHRNPC1
SCHEMBL14965737 0.88 CHRM1 (0.49) ALDH1A1TSHRMLLT1HDAC4KCNH2
SCHEMBL14965754 0.88 TSHR (0.47) ALDH1A1MEN1KMT2ATSHRMLLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed