SCHEMBL14965622

SCHEMBL14965622

O=C(CN1CCOc2nc([N+](=O)[O-])cn2CC1)NCc1ccc(-c2ccc(OC(F)(F)F)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.50
KCNH2 Q12809 4/20 0.47
GAA P10253 1/20 0.40
KMT2A Q03164 3/20 0.39
PTGS1 P23219 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
MEN1 O00255 1/20 0.37
ATM Q13315 1/20 0.37
USP2 O75604 1/20 0.37
HTT P42858 1/20 0.37
KIT P10721 1/20 0.37
ENPP2 Q13822 1/20 0.37
WNT3A P56704 1/20 0.36
SCN5A Q14524 1/20 0.36
SCN9A Q15858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965548 0.98 CHRM1 (0.52) CHRM1KCNH2GAAKMT2APTGS1
SCHEMBL14965849 0.88 CHRM1 (0.44) CHRM1KCNH2USP2HTT
SCHEMBL14965373 0.87 CA1 (0.48) KMT2AMEN1USP2HTT
SCHEMBL14966219 0.87 CA1 (0.48) CHRM1KCNH2KMT2AUSP2HTT
SCHEMBL14965804 0.86 KMT2A (0.41) CHRM1KCNH2KMT2AMEN1USP2
SCHEMBL14965624 0.86 CHRM1 (0.57) CHRM1KCNH2PTGS1SLC6A2SLC6A4
SCHEMBL14965737 0.85 CHRM1 (0.49) CHRM1KCNH2
SCHEMBL14966217 0.85 CHRM1 (0.50) CHRM1KCNH2GAAKMT2APTGS1
SCHEMBL14965565 0.84 KMT2A (0.43) KMT2AMEN1USP2HTT
SCHEMBL14965365 0.84 CHRM1 (0.49) CHRM1KCNH2KMT2APTGS1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed