SCHEMBL14965866

SCHEMBL14965866

O=[N+]([O-])c1cn2c(n1)OCCN(Cc1cncc(-c3cccc(F)c3)c1)CC2

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.42
DRD4 P21917 8/20 0.42
DRD3 P35462 8/20 0.42
HTR1A P08908 3/20 0.42
HTR2A P28223 1/20 0.42
HTR7 P34969 1/20 0.42
HTR2B P41595 1/20 0.42
DYRK1A Q13627 7/20 0.38
WNT1 P04628 1/20 0.38
CLK2 P49760 5/20 0.38
CLK3 P49761 5/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PLK4 O00444 1/20 0.35
GSK3B P49841 1/20 0.35
KLKB1 P03952 1/20 0.35
KLK1 P06870 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966131 0.92 DRD2 (0.49) DRD2DRD4DRD3HTR1AMEN1
SCHEMBL14965746 0.89 DRD2 (0.41) DRD2DRD4DRD3MEN1KMT2A
SCHEMBL14965749 0.85 CYP11B1 (0.43) DRD2DRD4DRD3MEN1KMT2A
SCHEMBL14965410 0.85 DRD2 (0.38) DRD2DRD4DRD3MEN1KMT2A
SCHEMBL14966240 0.85 KIT (0.40) DRD2DRD4DRD3
SCHEMBL14965957 0.84 DRD2 (0.40) DRD2DRD4DRD3HTR1AHTR2A
SCHEMBL14965683 0.84 DRD2 (0.43) DRD2DRD4DRD3HTR1AMEN1
SCHEMBL14971091 0.84 DRD2 (0.44) DRD2DRD4DRD3HTR1AMEN1
SCHEMBL14966205 0.83 LSS (0.46) DRD2DRD4DRD3HTR1A
SCHEMBL14965790 0.83 DRD2 (0.38) DRD2DRD4DRD3HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed