SCHEMBL14965749

SCHEMBL14965749

O=[N+]([O-])c1cn2c(n1)OCCN(Cc1ccc(-c3cccc(F)c3)nc1)CC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.43
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
STAT3 P40763 1/20 0.37
WNT3A P56704 2/20 0.36
MLNR O43193 4/20 0.36
PDE4B Q07343 1/20 0.36
MCHR1 Q99705 1/20 0.36
MET P08581 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.35
HSD17B10 Q99714 1/20 0.35
FLT3 P36888 1/20 0.34
TYRO3 Q06418 1/20 0.34
MERTK Q12866 1/20 0.34
GAS6 Q14393 1/20 0.34
SOS1 Q07889 1/20 0.34
CHRM1 P11229 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965746 0.89 DRD2 (0.41) DRD2DRD4DRD3PDE4BMEN1
SCHEMBL14965683 0.88 DRD2 (0.43) DRD2DRD4DRD3PDE4BMEN1
SCHEMBL14966131 0.88 DRD2 (0.49) DRD2DRD4DRD3PDE4BMEN1
SCHEMBL14965866 0.85 DRD2 (0.42) DRD2DRD4DRD3MEN1KMT2A
SCHEMBL14965805 0.85 DHODH (0.36) CYP11B1STAT3MCHR1METCHRM1
SCHEMBL14965730 0.85 DRD2 (0.37) DRD2DRD4DRD3PDE4BMEN1
SCHEMBL14965410 0.84 DRD2 (0.38) DRD2DRD4DRD3MEN1KMT2A
SCHEMBL14965932 0.84 HIF1A (0.41) STAT3CHRM1
SCHEMBL14965820 0.82 JAK2 (0.37) STAT3METMEN1KMT2AALDH1A1
SCHEMBL14965652 0.82 GPR119 (0.38) CYP11B1MLNRMCHR1MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed