SCHEMBL14966348

SCHEMBL14966348

CC1CCCc2cc(C(=O)O)c(N)nc21

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.39
HRH3 Q9Y5N1 7/20 0.37
HRH2 P25021 5/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
RCE1 Q9Y256 1/20 0.36
TBK1 Q9UHD2 9/20 0.35
IKBKE Q14164 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14967025 0.89 HRH3 (0.34) KDM4EHRH3HRH2NPC1RAB9A
SCHEMBL8136170 0.80 SLC9A1 (0.39) KDM4ENPC1RAB9AALDH1A1HPGD
SCHEMBL1680507 0.72 KDM4E (0.58) KDM4ENPC1RAB9AALDH1A1HPGD
SCHEMBL7911308 0.70 SLC9A1 (0.37) KDM4EHRH3HRH2NPC1RAB9A
SCHEMBL7916696 0.70 KDM4E (0.50) KDM4ENPC1RAB9AALDH1A1HPGD
SCHEMBL9406603 0.70 HRH3 (0.42) KDM4EHRH3HRH2HSD17B10MAPT
Fumaric Acid SCHEMBL7912855 0.68 SMN1; SMN2 (0.33) KDM4ENPC1RAB9AALDH1A1MAPT
Maleic Acid SCHEMBL7912919 0.68 SMN1; SMN2 (0.33) KDM4ENPC1RAB9AALDH1A1MAPT
SCHEMBL10286354 0.68 HSD17B10 (0.36) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL1998766 0.67 SLC9A1 (0.39) KDM4ERAB9AALDH1A1HSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072882-A1 2 -AMINO- 1, 8 -NAPHTHYRIDINE-3 -CARBOXAMIDE DERIVATIVES AS ANTIMICROBIAL AGENTS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-23 WO disclosed