SCHEMBL14967460

SCHEMBL14967460

O=Cc1ccc(-c2ccc(O[C@H]3CC[C@H](C(=O)O)CC3)nc2)cc1F

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 19/20 0.60
KCNH2 Q12809 5/20 0.54
SOAT1 P35610 3/20 0.54
ADORA2A P29274 1/20 0.48
ERN1 O75460 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14967507 1.00 DGAT1 (0.60) DGAT1KCNH2SOAT1ADORA2AERN1
SCHEMBL14968206 0.90 DGAT1 (0.53) DGAT1KCNH2SOAT1ADORA2AERN1
SCHEMBL15073375 0.90 DGAT1 (0.48) DGAT1KCNH2SOAT1ADORA2AERN1
SCHEMBL15055252 0.87 DGAT1 (0.49) DGAT1KCNH2SOAT1ADORA2AERN1
SCHEMBL15055254 0.87 DGAT1 (0.49) DGAT1KCNH2SOAT1ADORA2AERN1
SCHEMBL15055224 0.83 DGAT1 (0.51) DGAT1KCNH2SOAT1ADORA2AERN1
SCHEMBL14971569 0.83 DGAT1 (0.51) DGAT1KCNH2SOAT1ADORA2AERN1
SCHEMBL14971619 0.80 DGAT1 (0.77) DGAT1KCNH2SOAT1ADORA2A
SCHEMBL14971546 0.80 DGAT1 (0.42) DGAT1KCNH2SOAT1ADORA2AERN1
SCHEMBL14971566 0.80 DGAT1 (0.42) DGAT1KCNH2SOAT1ADORA2AERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013074387-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed