SCHEMBL15055252

SCHEMBL15055252

CCOC(=O)[C@H]1CC[C@@H](Oc2ccc(-c3ccc(C=O)c(F)c3)cn2)CC1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 16/20 0.49
KCNH2 Q12809 7/20 0.45
ADORA2A P29274 2/20 0.45
ERN1 O75460 1/20 0.43
SOAT1 P35610 4/20 0.42
ALDH1A1 P00352 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
PIK3CD O00329 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15055254 1.00 DGAT1 (0.49) DGAT1KCNH2ADORA2AERN1SOAT1
SCHEMBL14971562 0.89 DGAT1 (0.49) DGAT1KCNH2ADORA2AERN1SOAT1
SCHEMBL14971582 0.89 DGAT1 (0.41) DGAT1KCNH2ADORA2AERN1SOAT1
SCHEMBL14971557 0.89 DGAT1 (0.41) DGAT1KCNH2ADORA2AERN1SOAT1
SCHEMBL14967460 0.87 DGAT1 (0.60) DGAT1KCNH2ADORA2AERN1SOAT1
SCHEMBL14967507 0.87 DGAT1 (0.60) DGAT1KCNH2ADORA2AERN1SOAT1
SCHEMBL15073375 0.85 DGAT1 (0.48) DGAT1KCNH2ADORA2AERN1SOAT1
SCHEMBL14971566 0.85 DGAT1 (0.42) DGAT1KCNH2ADORA2AERN1SOAT1
SCHEMBL14971546 0.85 DGAT1 (0.42) DGAT1KCNH2ADORA2AERN1SOAT1
SCHEMBL15055224 0.82 DGAT1 (0.51) DGAT1KCNH2ADORA2AERN1SOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013096093-A1 COMPOUNDS AS DGAT-1 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-06-27 WO disclosed