SCHEMBL14969017

SCHEMBL14969017

NC(=O)c1cc2cc(C3CC3)c(C(F)(F)F)nc2nc1N

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.38
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 1/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
EEF2K O00418 3/20 0.34
SCN10A Q9Y5Y9 1/20 0.33
EEF2 P13639 1/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
MAPK1 P28482 1/20 0.31
SCN9A Q15858 2/20 0.31
TBK1 Q9UHD2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14969018 0.79 IKBKB (0.39) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL14966609 0.79 IKBKB (0.41) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL14969065 0.79 IKBKB (0.41) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL14968867 0.76 IKBKB (0.39) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL14968923 0.75 IKBKB (0.38) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL14969052 0.72 IKBKB (0.36) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL14969004 0.68 IKBKB (0.36) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL14968966 0.68 IKBKB (0.41) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL21905929 0.68 SCN10A (0.61) SCN10A
SCHEMBL14969024 0.68 RCE1 (0.36) IKBKBKDM4EALDH1A1GLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072882-A1 2 -AMINO- 1, 8 -NAPHTHYRIDINE-3 -CARBOXAMIDE DERIVATIVES AS ANTIMICROBIAL AGENTS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-23 WO claimed
WO-2013072882-A1 2 -AMINO- 1, 8 -NAPHTHYRIDINE-3 -CARBOXAMIDE DERIVATIVES AS ANTIMICROBIAL AGENTS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-23 WO disclosed