SCHEMBL14969415

SCHEMBL14969415

CC(C)NC(=O)c1ccc(-c2ccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.42
ALDH1A1 P00352 6/20 0.42
POLB P06746 1/20 0.41
LMNA P02545 2/20 0.41
CCR3 P51677 1/20 0.41
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
AURKA O14965 1/20 0.39
JAK2 O60674 1/20 0.39
JAK3 P52333 1/20 0.39
AURKB Q96GD4 1/20 0.39
MAPT P10636 2/20 0.39
CHKA P35790 1/20 0.39
KLKB1 P03952 1/20 0.38
KLK1 P06870 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14969456 0.97 POLB (0.43) ALDH1A1POLBLMNACCR3KMT2A
SCHEMBL14969471 0.92 KDM4E (0.41) ALDH1A1LMNAKMT2AMEN1MAPT
SCHEMBL14966204 0.89 SLC2A1 (0.42) ALDH1A1LMNAKMT2AMEN1AURKA
SCHEMBL14965848 0.88 MCHR1 (0.37) ALDH1A1KMT2AMEN1MCHR1
SCHEMBL14965741 0.88 MCHR1 (0.42) HDAC1HDAC6CHRM2MCHR1
SCHEMBL14965368 0.86 KCNJ1 (0.40) HRH3ALDH1A1LMNAKMT2AMEN1
SCHEMBL14966188 0.86 KDM4E (0.50) ALDH1A1CCR3KMT2AMEN1HDAC1
SCHEMBL14965370 0.86 ALDH1A1 (0.44) ALDH1A1LMNAKMT2AMEN1MAPT
SCHEMBL14971065 0.86 SLC2A1 (0.41) HRH3ALDH1A1LMNAKMT2AMEN1
SCHEMBL14965922 0.85 MAPT (0.46) ALDH1A1POLBLMNAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed